Deramciclane 对 <b>5-HT<sub>2A</sub></b> 和 <b>5-HT<sub>2C</sub></b> 受体具有高亲和力。Deramciclane 作为两种受体亚型的拮抗剂，对 5-HT<sub>2C</sub> 受体具有反向激动剂特性，无直接刺激激动剂。<BR><a href="https://www.medchemexpress.cn/GSK-2881078.html">GSK-2881078</a>产品描述：GSK 2881078 is a selective androgen receptor modulator potentially for the treatment of cachexia.
GSK 2881078 is a selective androgen receptor modulator (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting to improve their physical function.
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已为全球多个知名企业、院校构建各种定制型化合物库。</span><br><br>产品链接：<a href="http://www.medchemexpress.cn/GSK-2881078.html">www.medchemexpress.cn/GSK-2881078.html</a><br><br></span><img style="width: 600.0px;height: 310.0px;"
src="http://img.dxycdn.com/trademd/upload/userfiles/image/2014/08/A1408605159png_small.jpg"
alt="">Purity:98%<BR>MWt:301.4662<BR>Formula:C20H31NO<BR>SMILES:CC1(C)[C@]2(C)[C@@](OCCN(C)C)(C3=CC=CC=C3)C[C@@]1([H])CC2<BR>Pathway:GPCR/G Protein; Neuronal Signaling; <BR>Mechanisms:5-HT Receptor; <BR>Research Area:Neurological Disease<BR>电话： 021-58955995<BR>网址： www.MedChemExpress.cn <BR>地址： 上海市浦东新区蔡伦路720号2号楼3层
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